SCHEMBL6822902

SCHEMBL6822902

c1ccc(-c2nc[nH]c3nc4ccccc4c2-3)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
CYP3A4 P08684 4/20 0.49
MAPT P10636 4/20 0.49
PARP1 P09874 2/20 0.44
TNKS2 Q9H2K2 2/20 0.44
TNKS O95271 1/20 0.44
ADORA2A P29274 3/20 0.43
NUDT1 P36639 2/20 0.42
LMNA P02545 4/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA1 P30542 1/20 0.41
ALDH1A1 P00352 5/20 0.40
HPGD P15428 3/20 0.40
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
GAA P10253 4/20 0.40
HTT P42858 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2C9 P11712 3/20 0.40
CYP2C19 P33261 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2389719 0.78 GUSB (0.43) KDM4ECYP3A4MAPTPARP1TNKS2
SCHEMBL17047970 0.78 DCPS (0.43) KDM4ECYP3A4MAPTPARP1TNKS2
Hydrochloric Acid SCHEMBL7218019 0.77 GUSB (0.42) KDM4ECYP3A4MAPTPARP1TNKS2
SCHEMBL7216427 0.73 NPY5R (0.47) KDM4EALDH1A1HPGDSMN1; SMN2POLB
SCHEMBL5061741 0.72 LCK (0.42) KDM4ECYP3A4MAPTPARP1TNKS2
SCHEMBL2252074 0.70 ADORA2A (0.47) KDM4ECYP3A4MAPTADORA2ANUDT1
SCHEMBL971895 0.69 LMNA (0.62) KDM4ECYP3A4MAPTADORA2ANUDT1
SCHEMBL27810976 0.67 LMNA (0.61) KDM4ECYP3A4MAPTADORA2ANUDT1
SCHEMBL28239158 0.67 LMNA (0.61) KDM4ECYP3A4MAPTADORA2ANUDT1
SCHEMBL29514776 0.67 ESR1 (0.73) KDM4ECYP3A4MAPTADORA2ANUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058764-A1 4-PHENYL-PYRIMIDO [4,5-B] INDOLE DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-07-15 WO claimed
WO-2004058764-A1 4-PHENYL-PYRIMIDO [4,5-B] INDOLE DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-07-15 WO disclosed
WO-2004058764-A1 4-PHENYL-PYRIMIDO [4,5-B] INDOLE DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-07-15 WO disclosed