SCHEMBL6823710

SCHEMBL6823710

O=[N+]([O-])c1ccc(NC(=S)Nc2ccccc2)c(O)c1.O=[N+]([O-])c1ccc(NC(=S)Nc2ccccc2)c(O)c1

nearest known ligand 0.80

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.80
MAPT P10636 4/20 0.80
GAA P10253 2/20 0.80
HPGD P15428 2/20 0.80
CXCR1 P25024 4/20 0.73
CXCR2 P25025 4/20 0.73
SMN1; SMN2 Q16637 2/20 0.65
KCNMA1 Q12791 1/20 0.58
TDP1 Q9NUW8 2/20 0.57
NPC1 O15118 1/20 0.57
LMNA P02545 1/20 0.57
ALOX12 P18054 1/20 0.57
HTT P42858 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
HDAC6 Q9UBN7 1/20 0.55
KDM4E B2RXH2 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5594883 1.00 ALDH1A1 (0.80) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL7485596 0.95 CXCR2 (0.83) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL11674249 0.89 MAPT (1.00) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL28432107 0.86 ALDH1A1 (0.60) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL31222305 0.84 CXCR2 (1.00) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL5595180 0.84 CXCR2 (1.00) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL3708178 0.84 CXCR2 (0.79) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL5078630 0.82 ALDH1A1 (0.79) ALDH1A1MAPTGAAHPGDSMN1; SMN2
SCHEMBL28433444 0.82 RAB9A (0.72) ALDH1A1MAPTGAAHPGDCXCR1
SCHEMBL25250303 0.81 ALDH1A1 (0.60) ALDH1A1MAPTGAAHPGDCXCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1185261-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-02-25 EP disclosed
EP-1185261-A1 IL-8 RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-03-13 EP disclosed
WO-2000076495-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-21 WO disclosed