SCHEMBL6823744

SCHEMBL6823744

O=C(O)c1cccnc1N1CCN(c2ncc(C(=O)N3CCCC3)cc2Cl)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.48
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.46
CNR2 P34972 1/20 0.46
P2RY12 Q9H244 5/20 0.45
CXCR3 P49682 2/20 0.45
GRM5 P41594 1/20 0.44
HSD11B1 P28845 1/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HRH1 P35367 1/20 0.42
CCR3 P51677 1/20 0.42
KCNH2 Q12809 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7062607 0.82 CYP1A2 (0.58) KMT2APOLBGRM5HSD11B1ALDH1A1
SCHEMBL6826032 0.81 P2RY12 (0.49) POLBTSHRP2RY12CXCR3GRM5
SCHEMBL3309889 0.77 KMT2A (0.70) KMT2APOLBTSHRKDM4EALDH1A1
SCHEMBL11399275 0.75 KMT2A (0.68) KMT2APOLBTSHRCNR2KDM4E
SCHEMBL31057148 0.75 KMT2A (0.68) KMT2APOLBTSHRCNR2KDM4E
SCHEMBL17746092 0.75 KMT2A (0.68) KMT2APOLBTSHRKDM4EALDH1A1
SCHEMBL6919706 0.75 CYP2C9 (0.45) KMT2AP2RY12CXCR3GRM5HPGD
SCHEMBL13648884 0.75 CXCR3 (0.55) CXCR3HSD11B1
SCHEMBL6826225 0.75 HPGD (0.49) KMT2ATSHRCXCR3HPGDALDH1A1
Hydrochloric Acid SCHEMBL3976856 0.74 CXCR3 (0.54) CXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004074287-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-09-02 WO claimed
WO-2004074287-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-09-02 WO disclosed