SCHEMBL6823862

SCHEMBL6823862

CNc1nccc(-c2cc(C(=O)c3ccc(C)cc3F)ccc2O)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.42
JAK2 O60674 1/20 0.39
KDM1A O60341 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
CDK4 P11802 2/20 0.37
CDK2 P24941 1/20 0.37
HSD17B14 Q9BPX1 1/20 0.37
PDK1 Q15118 2/20 0.37
AKT3 Q9Y243 2/20 0.37
AURKA O14965 1/20 0.37
AURKB Q96GD4 1/20 0.37
TPX2 Q9ULW0 1/20 0.37
COMT P21964 1/20 0.37
RPS6KA3 P51812 1/20 0.36
CDKL1 Q00532 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826434 0.88 HDAC8 (0.39) HDAC8KDM1AHDAC1HDAC6HDAC2
SCHEMBL6826746 0.76 CDK1 (0.44) JAK2CDK2AKT3AURKBCOMT
SCHEMBL6826342 0.74 KMT2A (0.40) CDK2HSD17B14
SCHEMBL6824582 0.74 CYP46A1 (0.39) CDK2HSD17B14CYP19A1
SCHEMBL6823658 0.73 HSD17B14 (0.36) KDM1AHDAC1CDK2HSD17B14
SCHEMBL6824603 0.73 MAPT (0.39) CDK2HSD17B14RPS6KA3
SCHEMBL6917094 0.73 CDK2 (0.42) JAK2CDK4CDK2HSD17B14PDK1
SCHEMBL6823630 0.71 CDK1 (0.49) CDK2HSD17B14
SCHEMBL6824771 0.71 CDK1 (0.38) JAK2LOXL2CDK2HSD17B14AURKB
SCHEMBL6824151 0.71 IKBKB (0.34) KDM1AHDAC1LOXL2CDK2HSD17B14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed