SCHEMBL6824167

SCHEMBL6824167

Cc1ccc(C(=O)c2ccc(O)c(-c3cc(C(=O)NCCN4CCCC4)nc(N)n3)c2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ATR Q13535 1/20 0.42
CACNA1G O43497 5/20 0.41
SCN9A Q15858 4/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPK14 Q16539 1/20 0.40
KIT P10721 1/20 0.39
ABL1 P00519 1/20 0.39
MAP4K4 O95819 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824305 0.93 MAPK14 (0.48) MEN1KMT2AMAPK14
SCHEMBL6820704 0.81 CDK1 (0.59) MEN1KMT2AMAPK14KIT
SCHEMBL7064551 0.81 ADORA2A (0.41) ATRMEN1KMT2A
SCHEMBL6821420 0.79 CDK1 (0.43) MEN1KMT2AMAPK14
SCHEMBL6824731 0.79 ALDH1A1 (0.39) MEN1KMT2A
SCHEMBL6821385 0.78 MAPK14 (0.34) MAPK14KIT
SCHEMBL6823630 0.78 CDK1 (0.49)
SCHEMBL6923124 0.78 CDK1 (0.53) KMT2AMAPK14
SCHEMBL6824771 0.78 CDK1 (0.38) IKBKBMEN1KMT2A
SCHEMBL6823887 0.77 CDK2 (0.37) MEN1KMT2AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO claimed
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed