SCHEMBL6824355

SCHEMBL6824355

Cc1ccc(C(=O)c2ccc(O)c(-c3cc(NC(C)CN4CCOCC4)nc(N)n3)c2)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 2/20 0.42
CDK2 P24941 2/20 0.42
HDAC4 P56524 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
L3MBTL1 Q9Y468 3/20 0.37
MAPK14 Q16539 1/20 0.36
P2RX3 P56373 1/20 0.36
P2RX2 Q9UBL9 1/20 0.36
ABCB1 P08183 1/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALOX12 P18054 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6820704 0.86 CDK1 (0.59) CDK1CDK2MAPK14ALDH1A1HPGD
SCHEMBL6923124 0.85 CDK1 (0.53) CDK1CDK2L3MBTL1MAPK14ALDH1A1
SCHEMBL6824305 0.81 MAPK14 (0.48) CDK1CDK2MAPK14ALDH1A1HPGD
SCHEMBL6826440 0.81 CDK1 (0.55) CDK1CDK2ALDH1A1LMNAHPGD
SCHEMBL6824190 0.80 MAPK14 (0.43) CDK1CDK2L3MBTL1MAPK14ALDH1A1
SCHEMBL6826271 0.79 KDM4E (0.41) CDK1CDK2MAPK14ALDH1A1SMN1; SMN2
SCHEMBL6824361 0.79 MAPK14 (0.40) CDK1CDK2MAPK14ALDH1A1LMNA
SCHEMBL6826381 0.78 MAPK14 (0.39) CDK1CDK2L3MBTL1MAPK14ALDH1A1
SCHEMBL6824771 0.77 CDK1 (0.38) CDK1CDK2ALDH1A1HPGD
SCHEMBL6821420 0.77 CDK1 (0.43) CDK1CDK2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed