SCHEMBL6824812

SCHEMBL6824812

Cc1ccc(C(=O)c2ccc(OCc3ccccc3)c(-c3cc(NCCCN4CCOCC4)nc(N)n3)c2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.39
CDK2 P24941 1/20 0.39
NME2 P22392 2/20 0.39
TACR2 P21452 1/20 0.39
ERBB2 P04626 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 1/20 0.38
MC4R P32245 1/20 0.38
HSD17B10 Q99714 2/20 0.38
ALOX15 P16050 1/20 0.38
ROS1 P08922 1/20 0.38
ALK Q9UM73 1/20 0.38
MAPT P10636 3/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923124 0.86 CDK1 (0.53) CDK1CDK2ALDH1A1KMT2AROS1
SCHEMBL7068093 0.84 RAF1 (0.45) CDK1CDK2HSD17B10HPGDBRD4
SCHEMBL6820704 0.82 CDK1 (0.59) CDK1CDK2ALDH1A1KMT2AHSD17B10
SCHEMBL6821420 0.79 CDK1 (0.43) CDK1CDK2KMT2AMAPK14
SCHEMBL6823947 0.78 MRGPRX4 (0.43) BRD4
SCHEMBL6823543 0.77 MRGPRX4 (0.42) BRD4
SCHEMBL6916270 0.76 MRGPRX4 (0.41) KMT2ALMNAKDM4EMAPK1TDP1
SCHEMBL6826271 0.75 KDM4E (0.41) CDK1CDK2ALDH1A1PKMKDM4E
SCHEMBL6824190 0.73 MAPK14 (0.43) CDK1CDK2ALDH1A1KDM4EGAA
SCHEMBL6824305 0.73 MAPK14 (0.48) CDK1CDK2ALDH1A1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080979-A1 NOVEL 3-(2-AMINO-4-PYRIMIDINYL)-4-HYDROXYPHENYL KETONE DERIVATIVES LG LIFE SCIENCES LTD. (KR) 2004-09-23 WO disclosed