SCHEMBL6825099

SCHEMBL6825099

N#CCC1CCC2(CCN(Cc3ccccc3)CC2)O1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.61
OPRM1 P35372 2/20 0.49
CYP3A4 P08684 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824251 0.83 SIGMAR1 (0.58) SIGMAR1CYP3A4HSD17B10
SCHEMBL6773993 0.83 SIGMAR1 (0.58) SIGMAR1CYP3A4HSD17B10
SCHEMBL6823360 0.83 SIGMAR1 (0.59) SIGMAR1OPRM1CYP3A4HSD17B10
SCHEMBL6819672 0.80 SIGMAR1 (0.47) SIGMAR1
SCHEMBL6778524 0.76 SIGMAR1 (0.43) SIGMAR1CYP3A4HSD17B10
SCHEMBL3015327 0.73 SIGMAR1 (0.74) SIGMAR1
SCHEMBL2407205 0.73 CCR3 (0.65) SIGMAR1HRH3
SCHEMBL1966477 0.71 SIGMAR1 (0.61) SIGMAR1OPRM1CYP3A4HSD17B10
SCHEMBL6203773 0.70 DRD4 (0.66) SIGMAR1CYP3A4
SCHEMBL13548371 0.70 OPRM1 (0.60) SIGMAR1OPRM1CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058763-A1 4(SPIROPIPERIDINYL)METHYL SUBSTITUTED PYRROLIDINES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2004-07-15 WO disclosed