SCHEMBL6825655

SCHEMBL6825655

COC(=O)c1ccc(C=CC(=O)O)c(C)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
ATM Q13315 2/20 0.52
ESR1 P03372 2/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
XDH P47989 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
ITGB3 P05106 2/20 0.44
ITGAV P06756 2/20 0.44
ITGA2B P08514 2/20 0.44
ITGB1 P05556 1/20 0.44
ITGB5 P18084 1/20 0.44
NOTUM Q6P988 1/20 0.43
ALOX15 P16050 1/20 0.43
HTT P42858 1/20 0.43
ALDH1A1 P00352 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2827575 0.83 CTSL (0.54) KDM4EATMESR1TDP1ITGB3
SCHEMBL2824325 0.83 MIF (0.58) KDM4EATMCA12CA1CA2
SCHEMBL2827580 0.83 CTSL (0.54) KDM4EATMESR1TDP1ITGB3
SCHEMBL2824327 0.83 MIF (0.58) KDM4EATMCA12CA1CA2
SCHEMBL4316791 0.82 ESR1 (0.49) KDM4EESR1CA1CA2ITGB3
SCHEMBL4316794 0.82 ESR1 (0.49) KDM4EESR1CA1CA2ITGB3
SCHEMBL1496056 0.81 LCK (0.42) KDM4EATMESR1CA12CA1
SCHEMBL1496059 0.81 LCK (0.42) KDM4EATMESR1CA12CA1
SCHEMBL8702460 0.80 ALDH1A1 (0.57) KDM4EATMCA12CA1CA2
SCHEMBL8890648 0.80 ABCG2 (0.55) KDM4EATMCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487881-A2 SURFACE-ACTIVE PHOTOINITIATORS Ciba SC Holding AG (CH) 2004-12-22 EP disclosed
EP-1385912-A1 PYRIDONE DYES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE PRODUCTION OF COLOURED PLASTICS OR POLYMERIC COLOUR PARTICLES Ciba SC Holding AG (CH) 2004-02-04 EP disclosed
EP-1353959-A1 SURFACE-ACTIVE PHOTOINITIATORS Ciba SC Holding AG (CH) 2003-10-22 EP disclosed
EP-1335894-A2 BIS(ALKYLENEOXYBENZOPHENONE) ULTRAVIOLET LIGHT ABSORBERS CYTEC TECHNOLOGY CORP. (US) 2003-08-20 EP disclosed
WO-2003066687-A2 SURFACE-ACTIVE PHOTOINITIATORS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2003-08-14 WO disclosed
EP-1311627-A2 PROCESS FOR PRODUCING COATINGS USING SURFACE-ACTIVE PHOTOINITIATORS Ciba SC Holding AG (CH) 2003-05-21 EP disclosed
EP-1268047-A2 STERICALLY HINDERED PHENOL ANTIOXIDANT GRANULES HAVING BALANCED HARDNESS ALBEMARLE CORPORATION (US) 2003-01-02 EP disclosed
WO-2002090442-A1 PYRIDONE DYES, A PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE PRODUCTION OF COLOURED PLASTICS OR POLYMERIC COLOUR PARTICLES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2002-11-14 WO disclosed
WO-2002048204-A1 SURFACE-ACTIVE PHOTOINITIATORS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2002-06-20 WO disclosed
WO-2002046136-A2 BIS(ALKYLENEOXYBENZOPHENONE) ULTRAVIOLET LIGHT ABSORBERS CYTEC TECHNOLOGY CORP. (US) 2002-06-13 WO disclosed
WO-2002014439-A2 PROCESS FOR PRODUCING COATINGS USING SURFACE-ACTIVE PHOTOINITIATORS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2002-02-21 WO disclosed
WO-2001070869-A2 STERICALLY HINDERED PHENOL ANTIOXIDANT GRANULES HAVING BALANCED HARDNESS ALBEMARLE CORPORATION (US) 2001-09-27 WO disclosed
EP-1124832-A1 OXIME DERIVATIVES AND THE USE THEREOF AS LATENT ACIDS Ciba SC Holding AG (CH) 2001-08-22 EP disclosed
EP-1088027-A1 INCREASING THE MOLECULAR WEIGHT OF POLYESTERS Ciba SC Holding AG (CH) 2001-04-04 EP disclosed
WO-2000026219-A1 OXIME DERIVATIVES AND THE USE THEREOF AS LATENT ACIDS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2000-05-11 WO disclosed
WO-1999055772-A1 INCREASING THE MOLECULAR WEIGHT OF POLYESTERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-11-04 WO disclosed
US-4798822-A PHOTOSTABILIZERS FOR POLYMERS CIBA-GEIGY CORPORATION (US) 1989-01-17 US disclosed
US-4661594-A PHOTODEGRADATION INHIBITION CIBA-GEIGY CORPORATION (US) 1987-04-28 US disclosed