SCHEMBL6825815

SCHEMBL6825815

CCCOC(=O)CC(c1c(O)c2ccccc2oc1=O)C1CCCCC1.CCOC(=O)CC(c1c(O)c2ccccc2oc1=O)C1CCCC1.CCOC(=O)CC(c1c(O)c2ccccc2oc1=O)C1CCCCC1.COC(=O)CC(c1c(O)c2ccccc2oc1=O)C1CCCC1.O=C(O)CC(c1c(O)c2ccccc2oc1=O)C1CCCC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VKORC1 Q9BQB6 3/20 0.61
ADORA3 P0DMS8 1/20 0.48
NQO1 P15559 2/20 0.45
CYP2C9 P11712 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
ALB P02768 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PCSK7 Q16549 1/20 0.41
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CYP3A4 P08684 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CRHBP P24387 1/20 0.38
HTT P42858 1/20 0.38
CRHR2 Q13324 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6827896 0.93 VKORC1 (0.54) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL5106976 0.91 VKORC1 (0.73) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL5112793 0.90 VKORC1 (0.71) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL1647660 0.89 VKORC1 (0.76) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL5112806 0.88 VKORC1 (0.74) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL5100298 0.87 VKORC1 (0.78) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL5100246 0.86 VKORC1 (0.77) VKORC1ADORA3NQO1CYP2C9MEN1
SCHEMBL1648619 0.83 VKORC1 (0.81) VKORC1NQO1CYP2C9MEN1KMT2A
SCHEMBL6826370 0.83 VKORC1 (0.50) VKORC1CYP2C9MEN1KMT2AALDH1A1
SCHEMBL6827699 0.83 CYP2C9 (0.57) VKORC1ADORA3NQO1CYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383756-A1 COUMARIN DERIVATIVES TO BE USED AS ANTICOAGULANTS Arxy Therapeutics (US) 2004-01-28 EP disclosed
WO-2002085882-A1 COUMARIN DERIVATIVES TO BE USED AS ANTICOAGULANTS ARXY THERAPEUTICS (US) 2002-10-31 WO disclosed