SCHEMBL6826508

SCHEMBL6826508

CC(Cc1ccc(OC(F)(F)F)cc1)CC(C#N)C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.45
SLC6A4 P31645 2/20 0.40
EPHX1 P07099 1/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.38
EPHX2 P34913 2/20 0.37
PPARG P37231 2/20 0.37
PPARA Q07869 2/20 0.37
PDE2A O00408 1/20 0.36
SCN10A Q9Y5Y9 3/20 0.36
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
ALOX15 P16050 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4656296 0.84 ACACB (0.45) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL18012430 0.78 ACACB (0.48) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL5668779 0.76 ACACB (0.50) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL1912504 0.76 ACACB (0.51) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL23095147 0.75 ACACB (0.46) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL6825071 0.75 DAO (0.41) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL6824601 0.74 SLC6A2 (0.48) ACACBSLC6A4ALDH1A1KMT2ASLC6A2
SCHEMBL20821070 0.73 ACACB (0.49) ACACBSLC6A4EPHX1ALDH1A1TSHR
SCHEMBL14478297 0.73 SLC6A4 (0.61) ACACBSLC6A4EPHX1SCN10ASLC6A2
SCHEMBL14478239 0.73 SLC6A4 (0.61) ACACBSLC6A4EPHX1SCN10ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392647-A1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-03-03 EP disclosed
EP-1385817-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-02-04 EP disclosed
EP-1385377-A1 PESTICIDE COMPOSITION COMPRISING MALONONITRILE COMPOUNDS SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2004-02-04 EP disclosed
WO-2002090321-A1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed
WO-2002089579-A1 PESTICIDE COMPOSITION COMPRISING MALONONITRILE COMPOUNDS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed
WO-2002090320-A2 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-11-14 WO disclosed