SCHEMBL6833494

SCHEMBL6833494

NCc1ccc(NC(N)=S)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
TP53 P04637 1/20 0.56
TYR P14679 1/20 0.56
TSHR P16473 1/20 0.56
TAS2R38 P59533 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
ALOX12 P18054 1/20 0.55
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 2/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
KIF11 P52732 1/20 0.47
PLAU P00749 2/20 0.46
CYP1A2 P05177 1/20 0.46
ABAT P80404 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27517715 0.98 ALDH1A1 (0.54) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL16193023 0.84 MAPT (0.54) ALDH1A1TAS2R38HSD17B10CYP3A4CYP2C19
SCHEMBL16024387 0.84 ALDH1A1 (0.58) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL725810 0.83 ALDH1A1 (0.75) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL28701548 0.83 ALDH1A1 (0.56) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL2300811 0.81 GRIN2D (0.58) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL27295444 0.80 KMT2A (0.59) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL1893556 0.79 ALDH1A1 (0.52) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL28253803 0.79 CA2 (0.53) ALDH1A1ALOX12GAAMAPTPLAU
SCHEMBL27602582 0.79 IDO1 (0.60) ALDH1A1KMT2AGAAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1572299-A Medicine for improving excretion capacity of bladder TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2005-02-02 CN claimed
CN-107629022-A A kind of Trimethoprim and its preparation method and purposes 上海医药工业研究院 2018-01-26 CN disclosed
CN-107625766-A A kind of thiazole compound is used as the purposes of Trimethoprim 上海医药工业研究院 2018-01-26 CN disclosed
CN-107266388-A A kind of aminothiazole analog derivative 重庆大学 2017-10-20 CN disclosed
CN-104093701-B Separation method 旭化成株式会社 2017-05-03 CN disclosed
CN-101129295-B There is the binary initiator system of good storage stability and especially suitable for acidic system HERAEUS KULZER GMBH (DE) 2016-02-10 CN disclosed
CN-104093701-A Separation method ASAHI KASEI CHEMICALS CORP 2014-10-08 CN disclosed
CN-102367240-A 1,2,3-thiadiazole mother ring-contained iminothiazolone compounds, intermediate thereof, and preparation methods and applications of compound and intermediate UNIV EAST CHINA SCIENCE & TECH 2012-03-07 CN disclosed
CN-101277692-A Use of thiazole derivatives and analogues in the treatment of cancer BETAGENON AB (SE) 2008-10-01 CN disclosed
CN-100420678-C Cyclization process for substituted benzothiazole derivatives HOFFMANN LA ROCHE (CH) 2008-09-24 CN disclosed
CN-101237866-A Use of thiazole derivatives and analogues in the treatment of cancer BETAGENON AB (SE) 2008-08-06 CN disclosed
CN-101129295-A 2-component initiator system (amine free) with storage stability and especially suitable for acidic systems HERAEUS KULZER GMBH (DE) 2008-02-27 CN disclosed
CN-1738808-A Cyclization process for substituted benzothiazole derivatives HOFFMANN LA ROCHE (CH) 2006-02-22 CN disclosed
CN-1572299-A Medicine for improving excretion capacity of bladder TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2005-02-02 CN disclosed
EP-1467981-A1 4(HETERO-) ARYL SUBSTITUTED (THIA-/OXA-/PYRA) ZOLES FOR INHIBITION OF TIE-2 Kylix Pharmaceuticals B.V. (NL) 2004-10-20 EP disclosed
WO-2003062215-A1 4(HETERO-) ARYL SUBSTITUTED (THIA-/OXA-/PYRA) ZOLES FOR INHIBITION OF TIE-2 KYLIX PHARMACEUTICALS B.V. (NL) 2003-07-31 WO disclosed
CN-1035253-C Pyranyl cyanoguanidine derivatives SQUIBB & SONS INC (US) 1997-06-25 CN disclosed
CN-1064272-A PYRANYL CYANOGUANIDINE DERIVATIVES SQUIBB & SONS INC (US) 1992-09-09 CN disclosed
CN-86103798-A The preparation method of N-phenyl-4-phenyl-1-piperazine carbonamidine and their purposes as anti-arrhythmic 1987-06-10 CN disclosed