SCHEMBL6836592

SCHEMBL6836592

COc1ccc(-c2sc3cc(OC)ccc3c2C(=O)c2ccc(OCC3CCCCN3Cc3ccccc3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.60
ESR2 Q92731 16/20 0.60
ENPP3 O14638 2/20 0.51
ENPP1 P22413 2/20 0.51
CNR1 P21554 1/20 0.50
CNR2 P34972 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6836603 0.90 ESR1 (0.60) ESR1ESR2CNR1
SCHEMBL6601788 0.86 ESR1 (0.69) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL6601884 0.85 ESR1 (0.61) ESR1ESR2ENPP3ENPP1
SCHEMBL6600934 0.80 ESR1 (0.63) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL6836553 0.79 ESR1 (0.64) ESR1ESR2CNR1
SCHEMBL6600990 0.79 ESR1 (0.58) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL7452932 0.78 ESR1 (0.76) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL6604899 0.78 ESR1 (0.67) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL6602020 0.78 ESR1 (0.56) ESR1ESR2ENPP3ENPP1CNR1
SCHEMBL6603713 0.77 ESR1 (0.61) ESR1ESR2ENPP3CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6756388-B1 HAVING PIPERIDINYL AND PHENOLIC FUNCTIONALITY; BONE LOSS; BREAST OR PROSTATE CANCER PFIZER INC. 2004-06-29 US disclosed
EP-0723537-A1 BENZOTHIOPHENES AND RELATED COMPOUNDS AS ESTROGEN AGONISTS PFIZER INC. (US) 1996-07-31 EP disclosed
WO-1995010513-A1 BENZOTHIOPHENES AND RELATED COMPOUNDS AS ESTROGEN AGONISTS PFIZER INC. (US) 1995-04-20 WO disclosed