SCHEMBL6837441

SCHEMBL6837441

O=c1c([N+](=O)[O-])c(O)ccn1Cc1ccccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 8/20 0.46
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
HTT P42858 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 2/20 0.44
MAP3K14 Q99558 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.41
NPC1 O15118 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13120826 0.84 ALDH1A1 (0.45) PTGER3ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL3188133 0.83 HTT (0.52) ALDH1A1KDM4ESMN1; SMN2HTTLMNA
SCHEMBL8474847 0.82 PTGER3 (0.52) PTGER3ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL13120885 0.80 ALDH1A1 (0.37) ALDH1A1KDM4ESMN1; SMN2HTTL3MBTL1
SCHEMBL13120883 0.80 ALDH1A1 (0.38) ALDH1A1KDM4ESMN1; SMN2HTTL3MBTL1
SCHEMBL8486843 0.80 PTGER3 (0.44) PTGER3ALDH1A1SMN1; SMN2HTTLMNA
SCHEMBL14302460 0.78 PTGER3 (0.52) PTGER3ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL13120806 0.78 LMNA (0.51) PTGER3ALDH1A1KDM4ESMN1; SMN2HTT
SCHEMBL13120787 0.76 KMT2A (0.46) PTGER3ALDH1A1HTTL3MBTL1LMNA
SCHEMBL1770083 0.76 EGLN1 (0.62) PTGER3ALDH1A1KDM4ESMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
US-7812038-B2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
US-7812038-B2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS, INC. (US) 2010-10-12 US disclosed
EP-1176956-B1 CARBOXYLIC ACID DERIVATIVES THAT INHIBIT THE BINDING OF INTEGRINS TO THEIR RECEPTORS ENCYSIVE PHARMACEUTICALS INC (US) 2008-01-09 EP disclosed