SCHEMBL6840776

SCHEMBL6840776

COC(=O)[C@@H](N)CSc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
KIF11 P52732 1/20 0.42
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
GRM2 Q14416 1/20 0.39
THRB P10828 1/20 0.38
HTT P42858 1/20 0.38
HPGD P15428 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2951317 0.82 KIF11 (0.55) KIF11KMT2ARAB9A
SCHEMBL10977541 0.82 KIF11 (0.55) KIF11KMT2ARAB9A
Hydrochloric Acid SCHEMBL3610046 0.80 KIF11 (0.53) KIF11KMT2ARAB9A
Hydrochloric Acid SCHEMBL3610043 0.80 KIF11 (0.53) KIF11KMT2ARAB9A
SCHEMBL1693107 0.77 ALDH1A1 (0.49) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
SCHEMBL29627252 0.77 ALDH1A1 (0.49) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
SCHEMBL19699200 0.77 ALDH1A1 (0.49) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
SCHEMBL2058766 0.77 ALDH1A1 (0.49) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
Hydrochloric Acid SCHEMBL23824596 0.75 ALDH1A1 (0.48) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E
Hydrochloric Acid SCHEMBL5568685 0.75 ALDH1A1 (0.48) ALDH1A1KMT2ASMN1; SMN2GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6765109-B1 FORMATION OF ENANTIOSELECTIVE MATERIAL; REACTING ARYL THIOL AND PROTECTED SERINE DERIVATIVE ROCHE COLORADO CORPORATION 2004-07-20 US disclosed
EP-0968997-B1 Process for S-aryl-L-cysteine and derivatives HOFFMANN LA ROCHE (CH) 2003-10-01 EP disclosed
EP-1236715-A2 Process for S-Aryl cysteine F. HOFFMANN-LA ROCHE AG (CH) 2002-09-04 EP disclosed
US-6229041-B1 COUPLING CYSTEINE WITH COPPER OR COPPER OXIDE TO GENERATE METAL-AMINO COMPLEX, THEN CONTACTING WITH ARYL-HALIDE TO PRODUCE 3-ARYL-CYSTEINE; XENOBIOTIC METABOLIC PATHWAYS; TARGETTING HIV VIRUS F. HOFFMANN-LA ROCHE AG (CH) 2001-05-08 US disclosed
EP-0968997-A2 Process for S-aryl-L-cysteine and derivatives F. HOFFMANN-LA ROCHE AG (CH) 2000-01-05 EP disclosed