SCHEMBL6841735

SCHEMBL6841735

CCNc1nc(NCc2cccc(I)c2)c2ncn([C@@H]3O[C@H](c4cc(CC)no4)[C@@H](OC=O)[C@H]3O)c2n1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 17/20 0.51
ADORA1 P30542 7/20 0.51
ADORA2A P29274 6/20 0.51
ADORA2B P29275 2/20 0.49
HTR2C P28335 1/20 0.49
PPARG P37231 1/20 0.49
HTR2B P41595 1/20 0.49
PPARD Q03181 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
MAPT P10636 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6841733 0.95 ADORA3 (0.49) ADORA3ADORA1ADORA2AADORA2BHTR2C
Formic Acid SCHEMBL6841731 0.91 ADORA3 (0.56) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL6839134 0.90 ADORA3 (0.60) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL6839836 0.82 ADORA3 (0.66) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL6839831 0.81 ADORA3 (0.54) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL6839781 0.80 ADORA3 (0.53) ADORA3ADORA1ADORA2AADORA2BHTR2C
Acetic Acid SCHEMBL6839833 0.79 ADORA3 (0.69) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL6839114 0.79 ADORA2A (0.52) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL6839834 0.78 ADORA3 (0.68) ADORA3ADORA1ADORA2AHTR2CPPARG
SCHEMBL7595823 0.77 ADORA1 (0.48) ADORA3ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762170-B1 ANTIINFLAMMATORY AGENTS INHIBIT LEUKOCYTE RECRUITMENT AND ACTIVATION AND ARE AGONISTS OF THE ADENOSINE 2A RECEPTOR; PENDANT ISOXAZOLE; REACTING A 2,6-DIAMINOPURINE WITH A 2-(3-SUBSTITUTED ISOXAZOL-5-YL)TETRAHYDROFURAN-3,4-DIOL SMITHKLINEBEECHAM CORPORATION 2004-07-13 US disclosed
EP-1051425-B1 2-(PURIN-9-yl)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-10-30 EP disclosed