SCHEMBL684244

SCHEMBL684244

Cc1nc2c(c(=O)n(C)c(=O)n2C)n1CCN(C)C

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.51
TSHR P16473 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.48
MAPK1 P28482 2/20 0.48
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
RECQL P46063 1/20 0.47
USP2 O75604 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 2/20 0.45
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
GAA P10253 1/20 0.45
MAOB P27338 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11391007 0.98 CYP2D6 (0.53) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
SCHEMBL682738 0.91 SMN1; SMN2 (0.55) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
SCHEMBL684250 0.90 SMN1; SMN2 (0.54) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
Hydrochloric Acid SCHEMBL11387347 0.90 SMN1; SMN2 (0.57) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
Hydrochloric Acid SCHEMBL11384920 0.89 SMN1; SMN2 (0.56) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
SCHEMBL683577 0.85 TSHR (0.51) SMN1; SMN2TSHRL3MBTL1MAPK1CYP2C19
Hydrochloric Acid SCHEMBL11398174 0.84 TSHR (0.50) SMN1; SMN2TSHRL3MBTL1MAPK1CYP2C19
SCHEMBL683574 0.84 TSHR (0.47) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1
SCHEMBL683540 0.84 TSHR (0.50) SMN1; SMN2TSHRL3MBTL1MAPK1CYP2C19
Hydrochloric Acid SCHEMBL11397208 0.83 TSHR (0.46) CYP2D6SMN1; SMN2TSHRL3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4299832-A Substituted theophylline compounds FISONS LIMITED (GB) 1981-11-10 US claimed
EP-0011399-A1 N-substituted theophyllines, processes for their preparation and pharmaceutical compositions containing them FISONS plc (GB) 1980-05-28 EP claimed
US-20110269717-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN BRAINCELLS INC. (US) 2011-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110269717-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN NGF, DCX, BDNF CYP2D6 4428/4885SMN1; SMN2 907/4885TSHR 1873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.