SCHEMBL6843640

SCHEMBL6843640

O=C(Cl)c1cccc2[nH]c(CCl)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.44
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
DHODH Q02127 2/20 0.41
CHEK1 O14757 1/20 0.40
PLK4 O00444 1/20 0.40
MAPK13 O15264 1/20 0.40
DYRK3 O43781 1/20 0.40
ROCK2 O75116 1/20 0.40
RPS6KA5 O75582 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
CHEK2 O96017 1/20 0.40
PIM1 P11309 1/20 0.40
PHKG2 P15735 1/20 0.40
PRKACA P17612 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CSNK1D P48730 1/20 0.40
CLK2 P49760 1/20 0.40
GSK3A P49840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6841606 0.88 KDM4E (0.56) PARP1KDM4EHPGDDHODH
Hydrochloric Acid SCHEMBL4885974 0.86 KDM4E (0.55) PARP1KDM4EHPGDDHODH
SCHEMBL6841122 0.86 PARP1 (0.61) PARP1DHODHPLK4MAPK13DYRK3
SCHEMBL6841804 0.82 PKN1 (0.57) PARP1KDM4ECHEK1PKN1PKN2
SCHEMBL7485575 0.80 CHEK1 (0.52) PARP1KDM4ECHEK1PRKD3MAP4K4
SCHEMBL4033463 0.79 PARP1 (0.43) PARP1KDM4EHPGDCHEK1PKN1
SCHEMBL4066021 0.77 GRIN1 (0.54) PARP1KDM4ECHEK1
SCHEMBL4713439 0.76 TSHR (0.52) PARP1KDM4EHPGDCHEK1PKN1
SCHEMBL2307747 0.75 PSMB8 (0.53) PARP1CHEK1
SCHEMBL6582523 0.74 DDAH1 (0.42) KDM4ECHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040034078-A1 Benzimidazole inhibitors of poly(ADP-ribosyl) polymerase AGOURON PHARMACEUTICALS, INC. 2004-02-19 US disclosed
WO-2003106430-A1 BENZIMIDAZOLE INHIBITORS OF POLY(ADP-RIBOSYL) POLYMERASE PFIZER INC. (US) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040034078-A1 Benzimidazole inhibitors of poly(ADP-ribosyl) polymerase PARP1, PARP11, PARP2 PARP1 1/4885KDM4E 2460/4885HPGD 885/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.