SCHEMBL6844006

SCHEMBL6844006

COc1ccc([C@H](Br)C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
ALDH1A1 P00352 1/20 0.56
ACP3 P15309 1/20 0.53
LDHA P00338 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
AKR1C3 P42330 6/20 0.50
AKR1C2 P52895 6/20 0.50
PTGS2 P35354 3/20 0.50
PTGS1 P23219 3/20 0.50
CES2 O00748 3/20 0.50
CES1 P23141 3/20 0.50
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
PAX8 Q06710 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CDC42 P60953 1/20 0.50
RAC1 P63000 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL983848 1.00 CYP1A2 (0.56) CYP1A2ALDH1A1ACP3LDHAL3MBTL1
SCHEMBL8933321 0.84 ALDH1A1 (0.47) CYP1A2ALDH1A1ACP3L3MBTL1CES2
SCHEMBL7017619 0.84 ALDH1A1 (0.57) CYP1A2ALDH1A1ACP3L3MBTL1PTGS2
SCHEMBL11778400 0.84 AKR1C3 (0.69) CYP1A2L3MBTL1AKR1C3AKR1C2PTGS2
SCHEMBL378101 0.82 KMT2A (0.49) CYP1A2ALDH1A1CES2CES1NPC1
SCHEMBL7473317 0.82 PARP10 (0.52) CYP1A2ALDH1A1ACP3CES2CES1
SCHEMBL11451243 0.81 MAPT (0.56) ALDH1A1CES2CES1MAPTTSHR
SCHEMBL3089210 0.81 ALDH1A1 (0.62) CYP1A2ALDH1A1CES2CES1NPC1
SCHEMBL6201289 0.80 ALDH1A1 (0.61) CYP1A2ALDH1A1ACP3L3MBTL1CES2
SCHEMBL11302672 0.80 SRD5A2 (0.56) PTGS1CES2CES1TSHRPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6770775-B2 REACTING ACID HALIDES WITH A CINCHONA ALKALOID CATALYST AND A BASE TO FORM INTERMEDIATE KETENES, WHICH ARE THEN REACTED WITH ELECTROPHILIC HALOGENATING REAGENTS TO PRODUCE ALPHA-HALO-ESTERS WITH HIGH ENANTIOMERIC EXCESS WACK HARALD (DE) 2004-08-03 US claimed
US-6770775-B2 REACTING ACID HALIDES WITH A CINCHONA ALKALOID CATALYST AND A BASE TO FORM INTERMEDIATE KETENES, WHICH ARE THEN REACTED WITH ELECTROPHILIC HALOGENATING REAGENTS TO PRODUCE ALPHA-HALO-ESTERS WITH HIGH ENANTIOMERIC EXCESS WACK HARALD (DE) 2004-08-03 US disclosed
US-20030050501-A1 Method of synthesizing optically enriched alpha-halo-esters, and product and composition therefrom WACK HARALD (DE) 2003-03-13 US disclosed
US-5374656-A Nervous system disorders, gastrointestinal disorders RHONE-POULENC RORER, S.A. (FR) 1994-12-20 US disclosed