SCHEMBL684448

SCHEMBL684448

O=CC1(c2ccccc2)CO1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
CYP2C9 P11712 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
AKR1C1 Q04828 1/20 0.33
CHRNB2 P17787 1/20 0.33
SLC6A2 P23975 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2A6 P11509 1/20 0.33
OPRM1 P35372 3/20 0.32
OPRL1 P41146 2/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
OPRK1 P41145 1/20 0.32
CFTR P13569 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL10535963 0.98 MEN1 (0.33) MEN1CYP2C9KMT2ALMNAGAA
Water SCHEMBL11060484 0.98 MEN1 (0.33) MEN1CYP2C9KMT2ALMNAGAA
SCHEMBL7046139 0.86 NPC1 (0.30) CYP2C9
SCHEMBL7772327 0.77 LMNA (0.37) KMT2ALMNAGAACHRNB2SLC6A2
Water SCHEMBL11125328 0.77 SLC6A2 (0.38) CHRNB2SLC6A2CHRNB4CHRNA3CHRNA4
SCHEMBL136565 0.74 HTR2A (0.41) CHRNB2SLC6A2CHRNB4CHRNA3CHRNA4
SCHEMBL9215817 0.71 GRIN1 (0.36) MEN1CYP2C9KMT2AAKR1C1ALDH1A1
SCHEMBL28570949 0.71 TSHR (0.37) MEN1CYP2C9KMT2AGAAAKR1C1
SCHEMBL28411325 0.68 MAPK1 (0.36) MEN1KMT2ALMNAGAAAKR1C1
SCHEMBL28760491 0.68 GRIN1 (0.34) MEN1CYP2C9KMT2AAKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0114567-B1 1-CARBONYL-1-PHENYL-2-AZOLYL-ETHANOL DERIVATIVES AS MICROBICIDES AND PLANT GROWTH REGULATORS AND THEIR INTERMEDIATES CIBA-GEIGY AG (CH) 1988-09-14 EP claimed
US-8063050-B2 Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors ARRAY BIOPHARMA INC. (US) 2011-11-22 US disclosed
US-20080051399-A1 HYDROXYLATED AND METHOXYLATED PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS ARRAY BIOPHARMA INC. 2008-02-28 US disclosed
JP-2004352709-A METHOD FOR PRODUCING 1-AZOLE-2-PHENYL -2, 3-PROPANEDIOL DERIVATIVE MITSUI CHEMICALS INC 2004-12-16 JP disclosed
EP-0114567-B1 1-CARBONYL-1-PHENYL-2-AZOLYL-ETHANOL DERIVATIVES AS MICROBICIDES AND PLANT GROWTH REGULATORS AND THEIR INTERMEDIATES CIBA-GEIGY AG (CH) 1988-09-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080051399-A1 HYDROXYLATED AND METHOXYLATED PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS AKT1, AKT2, AKT1S1 MEN1 1677/4885CYP2C9 1373/4885KMT2A 1884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.