SCHEMBL6844602

SCHEMBL6844602

CN1C(=O)CN(C2CCC(F)(F)C2)c2nc(Cl)ncc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 3/20 0.39
PLK1 P53350 4/20 0.38
PLK2 Q9NYY3 2/20 0.38
PIK3CA P42336 6/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
BRD4 O60885 2/20 0.34
BRDT Q58F21 2/20 0.34
ALK Q9UM73 1/20 0.33
PIK3R1 P27986 5/20 0.32
TTK P33981 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RPS6KA3 P51812 1/20 0.31
STK4 Q13043 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6844719 0.91 PRKDC (0.39) PRKDCPLK1PLK2PIK3CAPIK3CD
SCHEMBL2875624 0.84 PRKDC (0.47) PRKDCPLK1PIK3CAPIK3CDPIK3CB
SCHEMBL2543788 0.84 PLK1 (0.38) PLK1PLK2PIK3CABRD4BRDT
SCHEMBL2544712 0.84 PLK1 (0.38) PLK1PLK2PIK3CABRD4BRDT
SCHEMBL2543786 0.84 PLK1 (0.38) PLK1PLK2PIK3CABRD4BRDT
SCHEMBL6840359 0.82 PRKDC (0.45) PRKDCPLK1PIK3CAPIK3CDPIK3CB
SCHEMBL6844375 0.82 PRKDC (0.45) PRKDCPLK1PIK3CAPIK3CDPIK3CB
SCHEMBL6844511 0.79 PRKDC (0.57) PRKDCPLK1PIK3CAPIK3CDPIK3CB
SCHEMBL30030718 0.79 PRKDC (0.57) PRKDCPLK1PIK3CAPIK3CDPIK3CB
SCHEMBL3702601 0.78 PIK3R1 (0.34) PLK1PLK2PIK3CAPIK3R1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079118-A1 PTERIDINONES AS INHIBITORS OF POLO-LIKE KINASE ELAN PHARMACEUTICALS, INC (US) 2011-06-30 WO disclosed