SCHEMBL6845708

SCHEMBL6845708

Bc1cccc2c1NC(=O)C2=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.60
DAO P14920 2/20 0.60
BCHE P06276 2/20 0.60
NSD2 O96028 1/20 0.60
LIG1 P18858 1/20 0.55
CASP3 P42574 1/20 0.54
CASP2 P42575 1/20 0.54
CASP7 P55210 1/20 0.54
CASP6 P55212 1/20 0.54
CASP8 Q14790 1/20 0.54
MAOA P21397 3/20 0.47
MAOB P27338 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
GSK3B P49841 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CDC25B P30305 1/20 0.39
PARP1 P09874 1/20 0.38
TGM2 P21980 2/20 0.37
DNMT1 P26358 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29417367 0.75 CES1 (1.00) CES1DAOBCHENSD2LIG1
SCHEMBL3088689 0.75 DAO (1.00) CES1DAOBCHENSD2LIG1
SCHEMBL29836255 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL281604 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL505703 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL1247382 0.75 CES1 (1.00) CES1DAOBCHENSD2LIG1
SCHEMBL29440762 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL31244367 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL5332282 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1
SCHEMBL29506270 0.75 CES1 (0.60) CES1DAOBCHENSD2LIG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119704-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed
EP-1812388-B1 SULFONAMIDE PERI-SUBSTITUTED BICYCLICS FOR OCCLUSIVE ARTERY DISEASE DECODE GENETICS EHF (IS) 2011-02-23 EP disclosed