SCHEMBL6847418

SCHEMBL6847418

NCc1cc2ccc(O)cc2[c]n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABAT P80404 1/20 0.36
ENPP2 Q13822 1/20 0.36
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
NPC1 O15118 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
CYP1A2 P05177 1/20 0.31
TYR P14679 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30
KMT2A Q03164 1/20 0.30
F12 P00748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6841772 0.77 HTR2A (0.35) HTR2ACYP1A2
SCHEMBL28254806 0.66 ESR2 (0.50) HTR2AHTR2CHTR2BESR1ESR2
SCHEMBL1450911 0.64 MEN1 (0.38) NPC1ESR1ESR2CYP1A2TYR
SCHEMBL28416019 0.63 ABAT (0.58) ABATENPP2ESR1ESR2CYP1A2
SCHEMBL2454279 0.63 ABAT (0.58) ABATENPP2ESR1ESR2CYP1A2
SCHEMBL5779818 0.62 ABAT (0.56) ABATENPP2ESR1ESR2CYP1A2
Benzylamine SCHEMBL5583890 0.61 ENPP2 (0.63) ABATENPP2NPC1ESR1ESR2
SCHEMBL23891903 0.59
SCHEMBL5827872 0.59 CYP1A2 (0.44) ESR1ESR2CYP1A2TYRF12
SCHEMBL12676044 0.58 MTNR1A (0.53) ABATENPP2ESR1ESR2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6768024-B1 CONTROLLING OBESITY, SEXUAL DYSFUNCTION OR INFLAMMATION LION BIOSCIENCE AG (DE) 2004-07-27 US claimed
WO-2002012166-A2 TRIAMINE DERIVATIVE MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME LION BIOSCIENCE AG (DE) 2002-02-14 WO claimed
US-6768024-B1 CONTROLLING OBESITY, SEXUAL DYSFUNCTION OR INFLAMMATION LION BIOSCIENCE AG (DE) 2004-07-27 US disclosed
WO-2002012166-A2 TRIAMINE DERIVATIVE MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME LION BIOSCIENCE AG (DE) 2002-02-14 WO disclosed