SCHEMBL6848110

SCHEMBL6848110

[CH2]C(c1cnc2ccccc2c1)C(C=O)c1cnc2ccccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
PDGFRB P09619 4/20 0.41
PDGFRA P16234 4/20 0.41
MGAM O43451 1/20 0.41
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 2/20 0.39
NQO1 P15559 1/20 0.39
KDM4E B2RXH2 2/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ACP1 P24666 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852009 0.78 NPC1 (0.45) ALDH1A1RAB9AKDM4EKMT2ASMN1; SMN2
SCHEMBL27720626 0.76 CYP1A2 (0.49) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL529903 0.76 CYP1A2 (0.44) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL12505007 0.75 PDGFRB (0.46) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL409414 0.74 CYP1A2 (0.42) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL4065530 0.74 CYP1A2 (0.48) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL5462379 0.73 CYP1A2 (0.44) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL15194838 0.71 NQO1 (0.43) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL29800505 0.70 CYP1A2 (0.44) CYP1A2PDGFRBPDGFRAMGAMALDH1A1
SCHEMBL372069 0.70 CYP1A2 (0.44) CYP1A2PDGFRBPDGFRAMGAMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1585775-A 6-O-acyl ketolide derivatives of erythromycine useful as antibacterials ORTHO MCNEIL PHARM INC (US) 2005-02-23 CN disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed