SCHEMBL6849953

SCHEMBL6849953

CN(C)C(c1ccc(CC(=O)O)cc1)n1c(=O)c2cc(Br)ccc2n2cnnc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
DNM1 Q05193 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TSHR P16473 1/20 0.32
MCL1 Q07820 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
QPCT Q16769 1/20 0.31
SRD5A2 P31213 1/20 0.31
TSPO P30536 1/20 0.31
OXER1 Q8TDS5 1/20 0.30
PTGS2 P35354 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6850185 0.93 SIRT1 (0.32) MAPTKDM4EDNM1SMN1; SMN2MCL1
SCHEMBL6854073 0.90 APEX1 (0.37) CYP26A1CYP3A4MAPTKDM4EALDH1A1
SCHEMBL6850091 0.86 PIK3R1 (0.31)
SCHEMBL6854433 0.83 PIK3R1 (0.36) HSD17B10SMN1; SMN2
SCHEMBL6850047 0.83 HPGD (0.32) MAPTKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6855394 0.78 SIGMAR1 (0.34) MEN1KMT2A
SCHEMBL6853742 0.74 SMN1; SMN2 (0.33) MAPTALDH1A1HPGDSMN1; SMN2TSHR
SCHEMBL6855372 0.74 CNR2 (0.32) ALDH1A1SMN1; SMN2MEN1KMT2AHTT
SCHEMBL6855687 0.74 CNR2 (0.33) HPGDSMN1; SMN2MEN1KMT2A
SCHEMBL6854194 0.73 APEX1 (0.36) MAPTKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6828315-B1 Anti- inflammatories, anti-allergics, bronchodilatators, anti-asthmatics, or TNF alpha inhibitors WARNER-LAMBERT LLC 2004-12-07 US claimed
US-6828315-B1 Anti- inflammatories, anti-allergics, bronchodilatators, anti-asthmatics, or TNF alpha inhibitors WARNER-LAMBERT LLC 2004-12-07 US disclosed
EP-1177195-B1 1-AMINO TRIAZOLO 4,3-a! QUINAZOLINE-5-ONES AND OR -5-THIONES INHIBITING PHOSPHODIESTERASE IV WARNER LAMBERT CO (US) 2003-03-19 EP disclosed