SCHEMBL6852216

SCHEMBL6852216

OC/C=C/c1ccc(-n2ccnn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 13/20 0.50
CYP19A1 P11511 1/20 0.44
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
RECQL P46063 1/20 0.39
KEAP1 Q14145 1/20 0.38
BRS3 P32247 1/20 0.33
KCNJ1 P48048 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852221 1.00 NOTUM (0.50) NOTUMCYP19A1ALDH1A1CYP3A4RECQL
SCHEMBL6850789 0.78 NOTUM (0.55) NOTUMCYP19A1ALDH1A1KEAP1KCNJ1
SCHEMBL6847993 0.77 ALDH1A1 (0.58) NOTUMALDH1A1CYP3A4RECQLBRS3
SCHEMBL6847991 0.77 ALDH1A1 (0.58) NOTUMALDH1A1CYP3A4RECQLBRS3
SCHEMBL10447781 0.76 NOTUM (0.78) NOTUMCYP19A1KEAP1BRS3
SCHEMBL6870749 0.75 NOTUM (0.51) NOTUMCYP19A1ALDH1A1KEAP1KCNJ1
SCHEMBL6870744 0.75 NOTUM (0.51) NOTUMCYP19A1ALDH1A1KEAP1KCNJ1
SCHEMBL6847715 0.75 NOTUM (0.51) NOTUMCYP19A1KEAP1
SCHEMBL6847717 0.75 NOTUM (0.51) NOTUMCYP19A1KEAP1
SCHEMBL6847719 0.75 NOTUM (0.51) NOTUMCYP19A1KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed