SCHEMBL6852558

SCHEMBL6852558

OCC=Cc1ccc(-c2ncno2)cc1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
ALDH1A1 P00352 1/20 0.39
RECQL P46063 1/20 0.39
KDM4E B2RXH2 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852553 1.00 CYP3A4 (0.39) CYP3A4ALDH1A1RECQLKDM4ECYP1A2
SCHEMBL6854147 0.78 KDM4E (0.33) CYP3A4KDM4ECYP1A2MAPTCYP2C9
SCHEMBL6847783 0.75 ALDH1A1 (0.43) CYP3A4ALDH1A1KDM4ECYP1A2MAPT
SCHEMBL6847776 0.75 ALDH1A1 (0.43) CYP3A4ALDH1A1KDM4ECYP1A2MAPT
SCHEMBL6879785 0.75
SCHEMBL6879790 0.75
SCHEMBL6848024 0.74 LTA4H (0.44) CYP3A4ALDH1A1RECQL
SCHEMBL6848028 0.74 LTA4H (0.44) CYP3A4ALDH1A1RECQL
SCHEMBL6850822 0.74 BRD4 (0.42) ALDH1A1KDM4EMAPT
SCHEMBL27594260 0.72 CA1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed