SCHEMBL6852609

SCHEMBL6852609

COc1nc(C(=O)N[C@@H]2CNC[C@H](O)C2)ccc1-n1cnc(C)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PSEN1 P49768 16/20 0.38
PSEN2 P49810 16/20 0.38
APH1B Q8WW43 16/20 0.38
NCSTN Q92542 16/20 0.38
APH1A Q96BI3 16/20 0.38
PSENEN Q9NZ42 16/20 0.38
CD38 P28907 1/20 0.37
BTK Q06187 2/20 0.36
APP P05067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852506 0.87 PSEN1 (0.38) NPC1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6854867 0.85 NPC1 (0.45) NPC1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6853649 0.81 CNR2 (0.40) NPC1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6852870 0.81 PSEN1 (0.57) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL155825 0.77 P2RX7 (0.46) CYP3A4CYP2C19PSEN1PSEN2APH1B
Hydrochloric Acid SCHEMBL194977 0.76 P2RX7 (0.45) CYP3A4CYP2C19PSEN1PSEN2APH1B
SCHEMBL9224077 0.76 MEN1 (0.51) CYP3A4CYP2C19PSEN1PSEN2APH1B
SCHEMBL6920437 0.76 USP30 (0.43) CYP3A4CYP2C19PSEN1PSEN2APH1B
Hydrochloric Acid SCHEMBL18527128 0.75 PSEN1 (0.44) CYP2C19PSEN1PSEN2APH1BNCSTN
SCHEMBL194967 0.74 PSEN1 (0.46) CYP3A4CYP2C19PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011059048-A1 NOVEL AMIDE DERIVATIVE 大日本住友製薬株式会社 (JP) 2011-05-19 WO disclosed