SCHEMBL6853005

SCHEMBL6853005

CCOC(=O)C=Cc1ccc(-c2ccc(C=CC(=O)O)cn2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.57
CA1 P00915 1/20 0.57
CA2 P00918 1/20 0.57
CA7 P43166 1/20 0.57
CA9 Q16790 1/20 0.57
CA14 Q9ULX7 1/20 0.57
TTR P02766 1/20 0.54
DPP4 P27487 1/20 0.54
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
HPGD P15428 2/20 0.52
MITF O75030 1/20 0.52
KLF5 Q13887 1/20 0.52
P4HTM Q9NXG6 1/20 0.51
CYP3A4 P08684 1/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
FDPS P14324 1/20 0.50
CASP3 P42574 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6853004 0.94 CA12 (0.64) CA12CA1CA2CA7CA9
SCHEMBL27792934 0.86 CA12 (0.75) CA12CA1CA2CA7CA9
SCHEMBL1579390 0.86 CA12 (0.75) CA12CA1CA2CA7CA9
SCHEMBL1579391 0.86 CA12 (0.75) CA12CA1CA2CA7CA9
SCHEMBL11076841 0.85 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL11076826 0.85 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL6853074 0.84 P4HTM (0.68) CA12CA1CA2CA7CA9
SCHEMBL29789035 0.84 P4HTM (0.68) CA12CA1CA2CA7CA9
SCHEMBL8731557 0.84 P4HTM (0.68) CA12CA1CA2CA7CA9
SCHEMBL8663795 0.82 CA12 (0.64) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799827-B1 ACRYLAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2004-05-12 EP disclosed
US-5786486-A ANTIMICROBIAL, ANTITUMOR AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1998-07-28 US disclosed
EP-0799827-A1 ACRYLAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-10-08 EP disclosed