SCHEMBL6853883

SCHEMBL6853883

[CH2]C#Cc1ccnc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.47
LOXL2 Q9Y4K0 1/20 0.44
HTR1A P08908 2/20 0.42
ADRA1D P25100 2/20 0.42
ADRA1A P35348 2/20 0.42
ADRA1B P35368 2/20 0.42
MAPT P10636 4/20 0.40
KDM4E B2RXH2 3/20 0.40
ADORA2A P29274 1/20 0.40
PTPN1 P18031 1/20 0.38
PTPN11 Q06124 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
CYP1A2 P05177 2/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15947627 0.88 NCF1 (0.54) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL6850673 0.87 MAPT (0.48) NCF1LOXL2MAPTKDM4EADORA2A
SCHEMBL15940574 0.83 ADORA2A (0.54) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL7207702 0.81 NCF1 (0.47) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL6851753 0.78 NCF1 (0.44) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL15947637 0.78 ACACB (0.44) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL21858037 0.78 ADORA2A (0.41) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL15940638 0.78 NCF1 (0.44) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL17370956 0.77 NCF1 (0.43) NCF1LOXL2HTR1AADRA1DADRA1A
SCHEMBL15940617 0.77 NCF1 (0.43) NCF1LOXL2HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1585775-A 6-O-acyl ketolide derivatives of erythromycine useful as antibacterials ORTHO MCNEIL PHARM INC (US) 2005-02-23 CN disclosed
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed