SCHEMBL6854128

SCHEMBL6854128

OCC(F)=Cc1ccc(-c2ncco2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 8/20 0.42
CHRNA7 P36544 1/20 0.37
CHRNA10 Q9GZZ6 1/20 0.37
CHRNA9 Q9UGM1 1/20 0.37
HPGDS O60760 1/20 0.36
HDAC4 P56524 2/20 0.36
KCNJ1 P48048 1/20 0.34
KCNH2 Q12809 1/20 0.34
ADRB3 P13945 1/20 0.33
BRD4 O60885 1/20 0.32
EDNRB P24530 1/20 0.31
EDNRA P25101 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6876954 1.00 LTA4H (0.42) LTA4HCHRNA7CHRNA10CHRNA9HPGDS
SCHEMBL6876949 1.00 LTA4H (0.42) LTA4HCHRNA7CHRNA10CHRNA9HPGDS
SCHEMBL6851810 0.81 LTA4H (0.44) LTA4HCHRNA7CHRNA10CHRNA9HPGDS
SCHEMBL6851804 0.81 LTA4H (0.44) LTA4HCHRNA7CHRNA10CHRNA9HPGDS
SCHEMBL6880729 0.76 NOTUM (0.51)
SCHEMBL6880734 0.76 NOTUM (0.51)
SCHEMBL6879779 0.76
SCHEMBL6879785 0.76
SCHEMBL6880725 0.76 NOTUM (0.51)
SCHEMBL6879790 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed
EP-1453847-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-09-08 EP disclosed
WO-2003050132-A1 6-O-ACYL KETOLIDE DERIVATIVES OF ERYTHROMYCINE USEFUL AS ANTIBACTERIALS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-06-19 WO disclosed