SCHEMBL6856152

SCHEMBL6856152

NS(=O)(=O)c1ccc(-n2nc(NC(=O)N=S)cc2-c2ccccc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.63
PTGS1 P23219 11/20 0.63
EPHX2 P34913 10/20 0.63
CA9 Q16790 4/20 0.58
CA1 P00915 3/20 0.58
CA2 P00918 3/20 0.58
PDPK1 O15530 1/20 0.55
CYP2C9 P11712 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6341958 0.86 PTGS2 (0.67) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL6350558 0.85 PTGS2 (0.66) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL6344713 0.85 PTGS2 (0.63) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL6757662 0.83 CA9 (0.66) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL8688440 0.81 PTGS2 (0.61) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL6353808 0.81 PTGS2 (0.70) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL9941537 0.80 CA9 (0.71) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL27517773 0.79 PTGS2 (0.64) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL8688495 0.79 PTGS2 (0.57) PTGS2PTGS1EPHX2CA9CA1
SCHEMBL5236666 0.77 RPA1 (0.72) PTGS2PTGS1EPHX2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6716991-B1 REACTING ETHYL DIFLUOROACETATE AND 4'-CHLOROACETOPHENONE PRODUCING 4,4-DIFLUORO-1-(4-(CHLORO)PHENYL)-BUTANE-1,3-DIONE AND REACTING WITH 4-SULPHONAMIDOPHENYL HYDRAZINE HYDROCHLORIDE G. D. SEARLE & CO. 2004-04-06 US disclosed