SCHEMBL6857313

SCHEMBL6857313

COc1cc(C=O)ccc1Oc1ccc(C(F)(F)F)cc1N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.57
RAB9A P51151 1/20 0.57
ALDH1A1 P00352 4/20 0.54
TSHR P16473 1/20 0.54
MAPT P10636 4/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TTR P02766 1/20 0.51
ESRRA P11474 6/20 0.48
FDPS P14324 1/20 0.48
CYP3A4 P08684 1/20 0.47
LMNA P02545 1/20 0.47
ATM Q13315 1/20 0.47
NQO2 P16083 1/20 0.43
HPGD P15428 2/20 0.43
AOX1 Q06278 1/20 0.43
TRIM24 O15164 1/20 0.43
ALDH5A1 P51649 1/20 0.43
ABAT P80404 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TRIM33 Q9UPN9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2699247 0.85 ESRRA (0.64) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL2382784 0.84 ESRRA (0.64) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL2382859 0.84 ESRRA (0.64) RAB9AALDH1A1TSHRMAPTTTR
SCHEMBL2380970 0.83 ESRRA (0.54) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL26936527 0.82 TTR (0.67) L3MBTL1RAB9AALDH1A1TSHRMAPT
SCHEMBL4262772 0.82 ALDH1A1 (0.51) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL2383238 0.81 ESRRA (0.66) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL2380688 0.81 ESRRA (0.66) ALDH1A1TSHRMAPTTTRESRRA
SCHEMBL399561 0.80 L3MBTL1 (0.66) L3MBTL1RAB9AALDH1A1TSHRMAPT
SCHEMBL5338649 0.80 ESRRA (0.59) ALDH1A1TSHRMAPTTTRESRRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2450352-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER Takeda Pharmaceutical Company Limited (JP) 2012-05-09 EP disclosed
WO-2011016501-A1 PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER 武田薬品工業株式会社 (JP) 2011-02-10 WO disclosed