SCHEMBL6858285

SCHEMBL6858285

O=C(O)CCCc1nc(NCc2ccc(O)c(Cl)c2)c2c(n1)sc1ccccc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.42
STAT6 P42226 2/20 0.41
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
HSD17B2 P37059 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
MAOB P27338 1/20 0.36
FFAR1 O14842 1/20 0.36
EGFR P00533 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6635949 0.97 HSD17B10 (0.41) HSD17B10STAT6CA1CA2HSD17B2
SCHEMBL6635468 0.97 HSD17B10 (0.41) HSD17B10STAT6CA1CA2HSD17B2
SCHEMBL6633539 0.95 HSD17B10 (0.43) HSD17B10STAT6CA1CA2HSD17B2
SCHEMBL6762774 0.93 TRPV1 (0.44) TRPV1MAOBFFAR1CYP1A2CYP2D6
SCHEMBL6853056 0.91 KDM4E (0.41) HSD17B10STAT6CA1CA2HSD17B2
SCHEMBL6219232 0.90 FFAR1 (0.43) TRPV1MAOBFFAR1
SCHEMBL6214624 0.90 FFAR1 (0.42) TRPV1MAOBFFAR1
SCHEMBL6860781 0.89 HSD17B10 (0.44) HSD17B10STAT6CA1CA2HSD17B2
SCHEMBL6762884 0.89 ACHE (0.45)
SCHEMBL6635736 0.89 STAT6 (0.42) HSD17B10STAT6CA1CA2HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6787548-B1 CARDIOVASCULAR INSUFFICIENCY AND ERECTILE DYSFUNCTION; 3-(4-(3-CHLORO-4-HYDROXYBENZYLAMINO) BENZO(4,5)THIENO(2,3-D)PYRIMIDIN-2-YL)PROPIONIC ACID MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2004-09-07 US disclosed