SCHEMBL6859397

SCHEMBL6859397

NC(=O)NC1CCN(Cc2ccc(Cl)cc2)C1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.61
DRD4 P21917 1/20 0.61
CCR2 P41597 12/20 0.61
TEAD1 P28347 1/20 0.59
GAA P10253 1/20 0.58
SIGMAR1 Q99720 1/20 0.57
BCHE P06276 1/20 0.56
ACHE P22303 1/20 0.56
BACE1 P56817 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27811320 0.87 DRD4 (0.67) DRD2DRD4SIGMAR1BCHEACHE
SCHEMBL27811321 0.87 DRD4 (0.67) DRD2DRD4SIGMAR1BCHEACHE
SCHEMBL22716940 0.87 DRD2 (0.66) DRD2DRD4CCR2TEAD1SIGMAR1
SCHEMBL4846218 0.86 CCR2 (0.65) DRD2DRD4CCR2TEAD1SIGMAR1
SCHEMBL4426840 0.86 CCR2 (0.65) DRD2DRD4CCR2TEAD1SIGMAR1
SCHEMBL4426833 0.86 CCR2 (0.65) DRD2DRD4CCR2TEAD1SIGMAR1
SCHEMBL4844836 0.84 CCR2 (0.71) DRD2DRD4CCR2SIGMAR1
SCHEMBL4847367 0.84 CCR2 (0.71) DRD2DRD4CCR2SIGMAR1
SCHEMBL4840672 0.83 CCR2 (0.57) DRD2DRD4CCR2TEAD1SIGMAR1
SCHEMBL4840662 0.83 CCR2 (0.57) DRD2DRD4CCR2TEAD1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1448566-A2 CHEMOKINE RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2004-08-25 EP disclosed
WO-2003045942-A2 CHEMOKINE RECEPTOR ANTAGONISTS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-06-05 WO disclosed