SCHEMBL6861858

SCHEMBL6861858

Cc1c(SCCOS(C)(=O)=O)ccnc1CNc1ncncc1Cl

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.31
CYP3A4 P08684 3/20 0.31
CYP2D6 P10635 3/20 0.31
CYP2C19 P33261 3/20 0.31
TSHR P16473 2/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862058 0.83 CYP1A2 (0.34) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6869025 0.76 CHRM4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6869763 0.74 SMN1; SMN2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6869698 0.74 CYP2D6 (0.44) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6865769 0.73 CHRM4 (0.33) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6867952 0.72 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6865865 0.72 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6866597 0.71 CYP1A2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6869900 0.69 CHRM4 (0.36) CYP1A2CYP3A4CYP2D6CYP2C19TSHR
SCHEMBL6871820 0.67 MAPT (0.36) CYP1A2CYP3A4CYP2D6CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091957-B1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA ALTANA PHARMA AG (DE) 2004-12-15 EP disclosed
US-6395732-B1 BACTERICIDES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2002-05-28 US disclosed
EP-1091957-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2001-04-18 EP disclosed
WO-1999061439-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1999-12-02 WO disclosed