SCHEMBL6869698

SCHEMBL6869698

Cc1c(SCCCN2CCNCC2)ccnc1CNc1ncncc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.44
CYP1A2 P05177 4/20 0.44
DRD3 P35462 2/20 0.37
DRD2 P14416 1/20 0.37
LMNA P02545 3/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
CYP3A4 P08684 4/20 0.33
HIF1A Q16665 2/20 0.33
CYP2C19 P33261 2/20 0.33
TSHR P16473 1/20 0.33
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
METAP1 P53582 7/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6865769 0.88 CHRM4 (0.33) CYP2D6CYP1A2LMNAKDM4EALDH1A1
SCHEMBL6862058 0.84 CYP1A2 (0.34) CYP2D6CYP1A2ALDH1A1CYP3A4HIF1A
SCHEMBL6861877 0.82 CYP1A2 (0.44) CYP2D6CYP1A2DRD3DRD2LMNA
SCHEMBL6861628 0.80 METAP1 (0.42) CYP2D6CYP1A2LMNAKDM4ENPC1
SCHEMBL6869025 0.77 CHRM4 (0.36) CYP2D6CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL7672106 0.76 DRD2 (0.39) CYP2D6CYP1A2DRD3DRD2LMNA
SCHEMBL6861858 0.74 CYP1A2 (0.31) CYP2D6CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL6869763 0.72 SMN1; SMN2 (0.39) CYP2D6CYP1A2LMNAKDM4ENPC1
Hydrochloric Acid SCHEMBL6861864 0.71 KDM4E (0.32) CYP2D6LMNAKDM4EALDH1A1CYP3A4
SCHEMBL6866116 0.69 METAP1 (0.33) CYP2D6DRD2LMNAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091957-B1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA ALTANA PHARMA AG (DE) 2004-12-15 EP disclosed
US-6395732-B1 BACTERICIDES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 2002-05-28 US disclosed
EP-1091957-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2001-04-18 EP disclosed
WO-1999061439-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1999-12-02 WO disclosed