SCHEMBL6861898

SCHEMBL6861898

COCc1cc(COC)cc(Nc2ccc(C#N)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.42
CYP2A6 P11509 1/20 0.40
KDR P35968 1/20 0.39
GSK3B P49841 1/20 0.39
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCG2 Q9UNQ0 7/20 0.38
ABCB1 P08183 6/20 0.38
DHODH Q02127 1/20 0.38
MAOB P27338 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ABCC1 P33527 2/20 0.37
ABCC3 O15438 1/20 0.37
ESR1 P03372 1/20 0.37
CYP1A2 P05177 1/20 0.37
PGR P06401 1/20 0.37
CHRM2 P08172 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL993599 0.78 CYP2A6 (0.58) EGLN2LOXL2CYP2A6MAOBKMT2A
SCHEMBL4694668 0.78 GRM5 (0.46) EGLN2LOXL2CYP2A6KDM4EMAOB
SCHEMBL395539 0.75 CA2 (0.52) LOXL2CYP2A6KDRSAE1UBA2
SCHEMBL5882916 0.75 F7 (0.41) EGLN2SAE1UBA2KDM4EMEN1
SCHEMBL20698865 0.74 GRM5 (0.46) EGLN2LOXL2CYP2A6KDM4EMAOB
SCHEMBL21042121 0.73 SAE1 (0.53) LOXL2CYP2A6KDRSAE1UBA2
SCHEMBL29470433 0.73 CSNK1D (0.61) GSK3BMEN1KMT2ACYP3A4ALDH1A1
SCHEMBL4124112 0.73 SAE1 (0.69) KDRSAE1UBA2KDM4EMEN1
SCHEMBL12736265 0.73 CYP2A6 (0.52) EGLN2LOXL2CYP2A6MAOBMAPT
SCHEMBL5612584 0.73 ALDH1A1 (0.52) CYP2A6KDRGSK3BABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149069-B1 PHENYLGLYCINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-25 EP disclosed