SCHEMBL6861935

SCHEMBL6861935

Cc1ccc(S(=O)(=O)N(C)c2ccc(O)c(C#N)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.58
MCOLN3 Q8TDD5 1/20 0.58
HTT P42858 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
ALDH1A1 P00352 1/20 0.47
LMNA P02545 3/20 0.47
C5AR1 P21730 1/20 0.44
BRD1 O95696 1/20 0.44
BRPF1 P55201 1/20 0.44
NR1H3 Q13133 2/20 0.43
GLA P06280 1/20 0.42
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
NR1H2 P55055 1/20 0.42
HCRTR2 O43614 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7077936 0.81 MAPT (0.67) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL2119843 0.80 MAPT (0.47) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL6863864 0.80 MEN1 (0.39) MAPTHTTNPSR1L3MBTL1ALDH1A1
SCHEMBL6864499 0.78 NR3C1 (0.57) MAPTNPSR1ALDH1A1LMNA
SCHEMBL2008337 0.75 MAPT (1.00) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL2117926 0.75 MAPT (0.50) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL2117920 0.75 MAPT (0.50) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL18031174 0.75 MAPT (0.82) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL6302212 0.75 MAPT (0.82) MAPTMCOLN3HTTNPSR1L3MBTL1
SCHEMBL2119973 0.73 MAPT (0.47) MAPTMCOLN3HTTNPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed