SCHEMBL6861964

SCHEMBL6861964

Cc1ccc(S(=O)(=O)N(Cc2ccccc2)c2ccc(OC[C@H](O)CNC(C)(C)CCCc3ccccc3)c(C#N)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.46
SLC6A2 P23975 5/20 0.46
SLC6A4 P31645 5/20 0.46
SLC6A3 Q01959 5/20 0.46
KCNH2 Q12809 5/20 0.46
CYP2D6 P10635 10/20 0.44
ADRB2 P07550 3/20 0.43
ALDH1A1 P00352 2/20 0.42
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
MAOA P21397 1/20 0.41
HTR2B P41595 1/20 0.41
ADRB3 P13945 1/20 0.41
NR3C1 P04150 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 1/20 0.39
SLC22A1 O15245 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861971 1.00 CASR (0.46) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6858010 0.96 CASR (0.47) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6858004 0.96 CASR (0.47) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6861996 0.88 CASR (0.44) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6862004 0.88 CASR (0.44) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6857683 0.86 CASR (0.60) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6863014 0.86 CASR (0.62) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6863019 0.86 CASR (0.62) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL6857684 0.86 CASR (0.60) CASRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL8168003 0.84 ALDH1A1 (0.45) ALDH1A1NR3C1LMNANPSR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP claimed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US claimed
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed