SCHEMBL6862801

SCHEMBL6862801

CN(C)CCOc1ncc(-c2ccc3ccccc3c2)c(C(=O)O)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.53
ALDH1A1 P00352 4/20 0.53
SMN1; SMN2 Q16637 1/20 0.42
CCNC P24863 4/20 0.41
CDK8 P49336 4/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
PAICS P22234 1/20 0.39
ESR1 P03372 1/20 0.39
TNKS O95271 1/20 0.39
LMNA P02545 1/20 0.39
CYSLTR1 Q9Y271 1/20 0.39
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
HTR1D P28221 1/20 0.38
POLB P06746 1/20 0.38
PIM1 P11309 1/20 0.38
PRKD3 O94806 1/20 0.38
PRKD1 Q15139 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylaminoethanol SCHEMBL6871396 0.96 ALDH1A1 (0.49) KDM4EALDH1A1SMN1; SMN2CCNCCDK8
SCHEMBL6871399 0.89 ALDH1A1 (0.48) KDM4EALDH1A1SMN1; SMN2CCNCCDK8
SCHEMBL6866149 0.83 KDM4E (0.44) KDM4EALDH1A1SMN1; SMN2PAICS
SCHEMBL6862186 0.81 HTR1B (0.47) KDM4EALDH1A1SMN1; SMN2CYSLTR1
SCHEMBL6866620 0.81 ALDH1A1 (0.44) KDM4EALDH1A1SMN1; SMN2POLB
SCHEMBL6862736 0.80 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2PAICS
SCHEMBL6862171 0.79 PIM1 (0.48) KDM4EALDH1A1CCNCCDK8PIM1
SCHEMBL6861974 0.79 HTR7 (0.56) KDM4EALDH1A1SMN1; SMN2
Dimethylaminoethanol SCHEMBL6868764 0.78 HTR1B (0.43) KDM4EALDH1A1SMN1; SMN2
SCHEMBL6872471 0.77 KDM4E (0.47) KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187814-B1 5-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-18 EP disclosed
US-6756380-B1 NEUROKININ 1 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. 2004-06-29 US disclosed
EP-1187814-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
WO-2000073278-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed