SCHEMBL6863310

SCHEMBL6863310

CCN(CC)C(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.64
F12 P00748 8/20 0.45
F2 P00734 6/20 0.45
PLAU P00749 2/20 0.43
PLG P00747 1/20 0.43
ATM Q13315 1/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6870656 0.93 ADORA2A (0.59) ADORA2AF12F2ATMALDH1A1
SCHEMBL6863726 0.93 ADORA2A (0.56) ADORA2AF12F2ALDH1A1LMNA
SCHEMBL6867223 0.93 ADORA2A (0.60) ADORA2AF12F2PLAUPLG
SCHEMBL6870369 0.91 ADORA2A (0.61) ADORA2AF12F2PLAUPLG
SCHEMBL6866841 0.91 ADORA2A (0.55) ADORA2AF12F2ATMALDH1A1
SCHEMBL6869794 0.89 ADORA2A (0.59) ADORA2AF12F2PLAUPLG
SCHEMBL6869823 0.89 ADORA2A (0.56) ADORA2AF12F2PLAUPLG
SCHEMBL6870680 0.88 ADORA2A (0.60) ADORA2AF12F2PLAUALDH1A1
SCHEMBL6868956 0.87 ADORA2A (0.59) ADORA2AF12F2PLAUPLG
SCHEMBL6871898 0.87 ADORA2A (0.62) ADORA2AF12F2PLAUPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed