SCHEMBL6869823

SCHEMBL6869823

CCCCN(CCC)C(=O)c1cc(N)n2nc(-c3ccccn3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.56
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
F12 P00748 7/20 0.40
F2 P00734 6/20 0.40
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
OPRK1 P41145 1/20 0.38
PLAU P00749 2/20 0.38
PLG P00747 1/20 0.38
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6867223 0.96 ADORA2A (0.60) ADORA2AHTR1ADRD2HTR2AF12
SCHEMBL6870656 0.94 ADORA2A (0.59) ADORA2AF12F2KDM4EGAA
SCHEMBL6873020 0.91 ADORA2A (0.53) ADORA2AF12F2KDM4EGAA
SCHEMBL6863310 0.89 ADORA2A (0.64) ADORA2AF12F2PLAUPLG
SCHEMBL6871898 0.87 ADORA2A (0.62) ADORA2AF12F2PLAUPLG
SCHEMBL6869475 0.87 ADORA2A (0.55) ADORA2AHTR1AHTR2AF12F2
SCHEMBL6872195 0.83 ADORA2A (0.55) ADORA2AF12F2PLAUPLG
SCHEMBL6870369 0.83 ADORA2A (0.61) ADORA2AF12F2PLAUPLG
SCHEMBL6863726 0.83 ADORA2A (0.56) ADORA2AF12F2KDM4EGAA
SCHEMBL6870680 0.82 ADORA2A (0.60) ADORA2AF12F2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1347974-B1 AMINOTRIAZOLOPYRIDIINE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed