SCHEMBL6863415

SCHEMBL6863415

CCOC(=O)Oc1oc2cccc(OCCCNCc3ccccc3)c2c1C

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NMT2 O60551 17/20 0.72
NMT1 P30419 17/20 0.72
ADRB2 P07550 2/20 0.49
ADRB1 P08588 2/20 0.49
ADRB3 P13945 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864133 0.90 NMT2 (0.59) NMT2NMT1ADRB2ADRB1ADRB3
SCHEMBL6874419 0.89 NMT2 (0.75) NMT2NMT1
SCHEMBL3471356 0.84 NMT2 (1.00) NMT2NMT1ADRB2ADRB1ADRB3
SCHEMBL6868611 0.83 NMT2 (0.64) NMT2NMT1
SCHEMBL6870237 0.82 NMT2 (0.70) NMT2NMT1ADRB2ADRB1ADRB3
Hydrochloric Acid SCHEMBL6869324 0.80 NMT2 (0.49) NMT2NMT1ADRB2ADRB1ADRB3
SCHEMBL6870479 0.80 NMT2 (0.76) NMT2NMT1
SCHEMBL6870905 0.80 MAOB (0.49) NMT2NMT1
SCHEMBL6868394 0.80 NMT2 (0.71) NMT2NMT1ADRB2ADRB1ADRB3
SCHEMBL6868285 0.79 NMT2 (0.72) NMT2NMT1ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379522-A1 DIHYDRO-BENZO(b)(1,4)DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS I F. HOFFMANN-LA ROCHE AG (CH) 2004-01-14 EP disclosed
WO-2002083665-A1 DIHYDRO-BENZO[b][1,4]DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS I F. HOFFMANN-LA ROCHE AG (CH) 2002-10-24 WO disclosed