SCHEMBL6863480

SCHEMBL6863480

FC(F)(F)c1cccc(CN2CCN(c3ccccc3)CC2)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.67
KDM4E B2RXH2 4/20 0.67
ALDH1A1 P00352 2/20 0.67
GAA P10253 2/20 0.67
POLB P06746 3/20 0.65
DRD4 P21917 1/20 0.64
HTR7 P34969 1/20 0.62
LMNA P02545 2/20 0.60
FAAH O00519 1/20 0.59
TSHR P16473 1/20 0.58
TP53 P04637 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
HTR1A P08908 1/20 0.56
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6862996 0.93 KDM4E (0.74) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL6864697 0.91 SIGMAR1 (0.76) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL15937919 0.88 HTR7 (0.69) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL5541643 0.88 DRD4 (0.63) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL5537735 0.88 KDM4E (0.62) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL5541635 0.88 KDM4E (0.62) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL11898006 0.86 KDM4E (0.70) SIGMAR1KDM4EALDH1A1GAAPOLB
SCHEMBL18965827 0.86 DRD4 (0.64) SIGMAR1KDM4EALDH1A1POLBDRD4
SCHEMBL7507938 0.85 SLC2A1 (0.58) SIGMAR1KDM4EPOLBDRD4HTR7
SCHEMBL6864524 0.85 KDM4E (0.68) SIGMAR1KDM4EALDH1A1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed
WO-1998005332-A1 NOVEL HETEROCYCLE COMPOSITIONS ISIS PHARMACEUTICALS, INC. (US) 1998-02-12 WO disclosed