SCHEMBL6863939

SCHEMBL6863939

CC(C)(N)Cc1cccc(Cl)c1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 3/20 0.57
TAAR1 Q96RJ0 3/20 0.52
IDO1 P14902 2/20 0.50
SLC6A2 P23975 2/20 0.44
HTR2A P28223 2/20 0.44
HTR2B P41595 2/20 0.44
SLC6A4 P31645 1/20 0.44
HRH1 P35367 1/20 0.44
CHRNA4 P43681 1/20 0.44
SLC6A3 Q01959 1/20 0.44
RECQL P46063 1/20 0.43
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
CYP2A13 Q16696 2/20 0.39
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
NR3C2 P08235 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30818122 1.00 PNMT (0.57) PNMTTAAR1IDO1SLC6A2HTR2A
Clortermine SCHEMBL164137 0.83 PNMT (0.52) PNMTTAAR1IDO1SLC6A2HTR2A
Clortermine SCHEMBL30295323 0.83 PNMT (0.52) PNMTTAAR1IDO1SLC6A2HTR2A
SCHEMBL6686200 0.83 PNMT (0.56) PNMTTAAR1IDO1SLC6A4ALDH1A1
Clortermine SCHEMBL266778 0.82 PNMT (0.50) PNMTTAAR1IDO1SLC6A2HTR2A
Clortermine SCHEMBL30791298 0.82 PNMT (0.50) PNMTTAAR1IDO1SLC6A2HTR2A
SCHEMBL30818163 0.80 PNMT (0.52) PNMTTAAR1IDO1SLC6A4ALDH1A1
SCHEMBL24776448 0.77 PNMT (0.48) PNMTTAAR1IDO1ALDH1A1KDM4E
SCHEMBL3909520 0.76 PNMT (0.47) PNMTTAAR1IDO1SLC6A4ALDH1A1
SCHEMBL9315343 0.75 PNMT (0.56) PNMTTAAR1IDO1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed