SCHEMBL6864124

SCHEMBL6864124

O=C(c1ccc(O)c(Cl)c1Cl)N1CCOCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.59
KDM4E B2RXH2 1/20 0.55
PHGDH O43175 1/20 0.53
HTT P42858 2/20 0.53
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA3 P07451 1/20 0.49
CA4 P22748 1/20 0.49
CA6 P23280 1/20 0.49
CA5A P35218 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA13 Q8N1Q1 1/20 0.49
CA14 Q9ULX7 1/20 0.49
CA5B Q9Y2D0 1/20 0.49
ERN1 O75460 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28744516 0.86 HSP90AA1 (0.55) HSP90AA1KDM4EPHGDHHTTMAPT
SCHEMBL23021686 0.79 KDM4E (0.61) HSP90AA1KDM4EPHGDHHTTMAPT
SCHEMBL487433 0.79 KDM4E (0.75) HSP90AA1KDM4EPHGDHHTTMAPT
SCHEMBL6862139 0.79 KMT2A (0.54) KDM4EHTTMAPTTSHRSMN1; SMN2
SCHEMBL18299399 0.76 ERN1 (0.58) HSP90AA1KDM4EPHGDHHTTMAPT
SCHEMBL18299935 0.76 KDM4E (0.57) HSP90AA1KDM4EHTTMAPTTSHR
SCHEMBL18299000 0.76 KDM4E (0.57) HSP90AA1KDM4EHTTMAPTTSHR
SCHEMBL4469583 0.75 TSHR (0.71) HSP90AA1KDM4EHTTMAPTTSHR
SCHEMBL29486100 0.75 GAA (0.52) HSP90AA1KDM4EPHGDHHTTMAPT
SCHEMBL28746378 0.75 GAA (0.52) HSP90AA1KDM4EPHGDHHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973730-B1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2004-06-16 EP disclosed
US-6294531-B1 AMINOALKANOLS AS BLOOD COAGULANTS SMITHKLINE BEECHAM CORPORATION 2001-09-25 US disclosed
EP-0973730-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2000-01-26 EP disclosed
WO-1998045255-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-15 WO disclosed