SCHEMBL6864563

SCHEMBL6864563

O=C(CN1CCN(Cc2cccc([N+](=O)[O-])c2)CC1)NO

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.65
KDM4E B2RXH2 6/20 0.65
MAPK1 P28482 2/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
NPSR1 Q6W5P4 1/20 0.65
LMNA P02545 3/20 0.63
POLB P06746 2/20 0.63
MAPT P10636 1/20 0.63
TDP1 Q9NUW8 1/20 0.60
L3MBTL1 Q9Y468 2/20 0.60
SIGMAR1 Q99720 1/20 0.57
FAAH O00519 1/20 0.56
MGLL Q99685 1/20 0.56
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
CYP2D6 P10635 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
RECQL P46063 1/20 0.54
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15800712 0.85 ALDH1A1 (0.78) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL6864897 0.85 ALDH1A1 (0.66) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL28215819 0.83 ALDH1A1 (0.68) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL6862228 0.83 SIGMAR1 (0.67) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL6864679 0.83 ALDH1A1 (0.58) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL15279117 0.82 CYP2D6 (0.63) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL14424712 0.82 CYP2D6 (0.63) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL29078396 0.81 CYP2C19 (0.59) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL2930608 0.81 ALDH1A1 (0.71) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1
SCHEMBL7859148 0.80 ALDH1A1 (0.69) ALDH1A1KDM4EMAPK1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed
US-6800444-B1 USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS/INTERMEDIATES ISIS PHARMACEUTICALS, INC. 2004-10-05 US disclosed
US-6660466-B1 Reacting reactive appendage compounds such as meta benzylic compounds or alpha-amide compounds with scaffold molecules having reactive functionalities and contacting the intermediate library with a reducing agent ISIS PHARMACEUTICALS, INC. 2003-12-09 US disclosed
US-6150129-A USEFUL AS ANTIBACTERIAL AND OTHER PHARMACEUTICAL AGENTS AND AS INTERMEDIATES FOR PREPARATION OF OTHER PHARMACEUTICAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 2000-11-21 US disclosed
US-5922872-A BACTERICIDES AND DRUGS ISIS PHARMACEUTICALS, INC. (US) 1999-07-13 US disclosed
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US disclosed
US-5798360-A ANTIBACTERIAL AGENTS ISIS PHARMACEUTICALS, INC. (US) 1998-08-25 US disclosed
US-5780241-A ALTERING ELECTROCHEMICAL PROPERTIES BY DECYCLIZATION ISIS PHARMACEUTICALS, INC. (US) 1998-07-14 US disclosed
WO-1998020349-A1 COMPLEX CHEMICAL LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-05-14 WO disclosed
US-5731438-A BACTERICIDES; DRUGS ISIS PHARMACEUTICALS, INC. (US) 1998-03-24 US disclosed