SCHEMBL6865786

SCHEMBL6865786

Cc1nc(C)c(Cl)c(NCc2nccc(OCCCCSCc3cccnc3)c2C)n1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NMT2 O60551 7/20 0.36
NMT1 P30419 7/20 0.36
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 3/20 0.36
HPGD P15428 1/20 0.35
PDE10A Q9Y233 1/20 0.35
SCN8A Q9UQD0 1/20 0.33
PGK1 P00558 1/20 0.33
CYP1A2 P05177 3/20 0.33
CYP3A4 P08684 3/20 0.33
CYP2D6 P10635 3/20 0.33
ALOX15 P16050 3/20 0.33
CYP2C19 P33261 3/20 0.33
HSD17B10 Q99714 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
PKM P14618 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044854 0.90 HPGD (0.32) HPGDPDE10A
SCHEMBL6869916 0.87 HPGD (0.32) HPGDPDE10A
SCHEMBL6872699 0.85 PDE10A (0.35) NMT2NMT1ALDH1A1KDM4EHPGD
SCHEMBL6866232 0.84 KCNH2 (0.38) ALDH1A1KDM4EPDE10ASCN8APGK1
SCHEMBL6861630 0.84 PDE10A (0.32) HPGDPDE10ACYP1A2CYP3A4CYP2D6
SCHEMBL6866284 0.83 KDM4E (0.35) ALDH1A1KDM4EHPGDPDE10APGK1
SCHEMBL6869856 0.83
SCHEMBL6870015 0.81 ALDH1A1 (0.43) ALDH1A1HPGDCYP1A2CYP2D6ALOX15
SCHEMBL6871021 0.81 PDE10A (0.30) PDE10A
SCHEMBL6861500 0.81 DYRK3 (0.33) ALDH1A1KDM4EHPGDPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091957-B1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA ALTANA PHARMA AG (DE) 2004-12-15 EP disclosed
EP-1091957-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 2001-04-18 EP disclosed
WO-1999061439-A1 PYRIMIDIN-AMINOMETHYL-PYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN THE CONTROL OF HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1999-12-02 WO disclosed