SCHEMBL6866448

SCHEMBL6866448

CN(C)CCN.Cc1ccccc1-c1cnc(NCCN(C)C)nc1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.41
ATM Q13315 1/20 0.39
ZAP70 P43403 1/20 0.38
PIK3CD O00329 1/20 0.36
CSNK2A1 P68400 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PRKDC P78527 1/20 0.35
ATR Q13535 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
FGFR1 P11362 2/20 0.35
ELANE P08246 1/20 0.35
POLB P06746 1/20 0.35
RAD52 P43351 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6869463 0.95 ATM (0.43) SYKATMPIK3CDCSNK2A1KDM4E
SCHEMBL6866685 0.88 RAD52 (0.39) SYKATMZAP70CSNK2A1POLB
SCHEMBL6868453 0.87 HTR7 (0.41) SYKATMKDM4EALDH1A1SMN1; SMN2
SCHEMBL6872231 0.86 NMT2 (0.41) SYKZAP70CSNK2A1
SCHEMBL6016404 0.84 SYK (0.45) SYKZAP70CSNK2A1ELANEPOLB
SCHEMBL6873419 0.83 PIM1 (0.45) SYKATMZAP70CSNK2A1KDM4E
SCHEMBL6869416 0.83 ATM (0.50) SYKATMCSNK2A1KDM4EALDH1A1
SCHEMBL6862593 0.82 KDM4E (0.46) SYKATMCSNK2A1KDM4EALDH1A1
SCHEMBL6862307 0.82 CSNK2A1 (0.43) SYKATMCSNK2A1KDM4EALDH1A1
SCHEMBL6866454 0.81 POLB (0.39) SYKPIK3CDKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187814-B1 5-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2004-08-18 EP disclosed
US-6756380-B1 NEUROKININ 1 RECEPTOR ANTAGONISTS HOFFMANN-LA ROCHE INC. 2004-06-29 US disclosed
EP-1187814-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
WO-2000073278-A2 5-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed